Queen's Award Received in 2021 ISO 9001 Certified Delivered over 1,000,000 bio-reagents to life science researchers Trusted by Life Science Communities
Cart summary

You have no items in your shopping cart.

ERα antagonist 1

SKU: orb1686014

Description

ERα antagonist 1 is a potent and selective covalent inhibitor of estrogen receptor alpha. It induces G0/G1 cell cycle arrest and apoptosis in ERα-positive breast cancer cells like MCF-7, making it a valuable tool for investigating ERα biology and therapeutic strategies in both cellular and animal models of hormone-dependent cancers.

Research Area

Cell Biology, Metabolism Research, Pharmacology & Drug Discovery

Images & Validation

Key Properties

CAS Number2762423-09-4
MW568.68
FormulaC33H32N2O5S
SMILESC(=O)(C1=C(SC=2C1=CC=C(O)C2)C3=CC=C(O)C=C3)C4=CC=C(OC5CN(C/C=C/C(=O)N6CCCCC6)C5)C=C4
TargetEstrogen Receptor/ERR,Others,Apoptosis

Storage & Handling

Storage-20°C
Expiration Date12 months from date of receipt.
DisclaimerFor research use only

Similar Products

  • Atopaxar Hydrobromide [orb1705932]

    >99.99% (May vary between batches)

    474550-69-1

    608.54

    C29H39BrFN3O5

    5 mg, 10 mg, 1 mg, 25 mg
  • Atopaxar [orb1705936]

    98.50% (May vary between batches)

    751475-53-3

    527.63

    C29H38FN3O5

    100 mg, 1 ml x 10 mM (in DMSO), 1 mg, 5 mg, 10 mg, 25 mg, 50 mg
  • PB28 [orb1704256]

    >98%

    172907-03-8

    443.5

    C24H38N2O·2HCl

    5 mg, 25 mg
  • G36 [orb1704521]

    99.86% (May vary between batches)

    1392487-51-2

    412.32

    C22H22BrNO2

    5 mg, 10 mg, 50 mg, 1 mg, 25 mg, 100 mg, 500 mg, 1 ml x 10 mM (in DMSO)
  • Giredestrant tartrate [orb1709734]

    >99.99% (May vary between batches)

    2407529-33-1

    672.64

    C31H37F5N4O7

    1 mg, 10 mg, 25 mg, 50 mg, 5 mg
Quality Guarantee

Quality Guarantee

Explore bioreagents carefree to elevate your research. All our products are rigorously tested for performance. If a product does not perform as described on its datasheet, our scientific support team will provide expert troubleshooting, a prompt replacement, or a refund. For full details, please see our Terms & Conditions and Buying Guide. Contact us at [email protected].

Key Properties

No computed properties available.

Protocol Information