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ETA antagonist 1

SKU: orb1709061

Description

ETA antagonist 1 is a selective endothelin receptor type A (ETA) antagonist with an IC50 of 80 nM. This small molecule inhibitor is a valuable research tool for studying the role of ETA in cardiovascular diseases, pulmonary hypertension, and cancer biology in both cellular and animal models.

Research Area

Pharmacology & Drug Discovery

Images & Validation

Key Properties

CAS Number161801-60-1
MW387.5
FormulaC20H25N3O3S
SMILESS(NC1=C(C)C(C)=NO1)(=O)(=O)C=2C3=C(C(NCCCCC)=CC=C3)C=CC2
TargetEndothelin Receptor,Others

Storage & Handling

Storage-20°C
Expiration Date12 months from date of receipt.
DisclaimerFor research use only

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Key Properties

No computed properties available.

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ETA antagonist 1 (orb1709061)

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Step 1: Enter information below

(Recommended: An additional animal making an allowance for loss during the experiment)

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