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Rapastinel

SKU: orb1226869

Description

A tetrapeptide (TPPT-amide) that acts as a NMDA receptor glycine site partial agonist; readily crosses the blood-brain barrier and modulates the NMDA receptor, shows potent cognitive-enhancing properties in a valid in vivo model of learning.Depression Phase 3 Clinical.

Images & Validation

Key Properties

CAS Number117928-94-6
MW413.4686
Purity>98% (HPLC)
FormulaC18H31N5O6
SMILESC[C@@H](O)[C@@H](C(N)=O)NC([C@H]1N(C([C@H]2N(C([C@H]([C@H](O)C)N)=O)CCC2)=O)CCC1)=O
TargetiGluR
SolubilityDMSO: ≥ 32 mg/mL

Storage & Handling

StorageStorage temperature: -20°C. Stability: ≥ 2 years
Expiration Date12 months from date of receipt.
DisclaimerFor research use only

Alternative Names

GLYX-13 | Thr-Pro-Pro-Thr-NH2

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Rapastinel (orb1226869)

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(Recommended: An additional animal making an allowance for loss during the experiment)

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% DMSO +
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% Tween 80 +
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Available Sizes

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100 mg
200 mg
500 mg
5 mg
$ 140.00
10 mg
$ 180.00
25 mg
$ 340.00
50 mg
$ 490.00