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PNU-282987

SKU: orb1305505

Description

PNU-282987

Research Area

Neuroscience, Pharmacology & Drug Discovery

Images & Validation

Key Properties

CAS Number123464-89-1
MW301.21
Purity99.97%
FormulaC14H18Cl2N2O
SMILESCl.C1CN2CCC1[C@H](C2)NC(=O)c1ccc(cc1)Cl
TargetAChR,5-HT Receptor
SolubilityH2O:25 mg/mL (83 mM);10% DMSO+90% Corn Oil:1.67 mg/mL (5.54 mM);DMSO:250 mg/mL (829.99 mM)

Bioactivity

Target IC50
α7 nAChR (rat):26 nM(Ki)

Storage & Handling

StoragePowder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature.
Expiration Date12 months from date of receipt.
DisclaimerFor research use only

Alternative Names

inhibit, nAChR, Nicotinic acetylcholine receptors, Inhibitor, α7 nAChR, PNU282987, PNU-282987, PNU 282987

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Quality Guarantee

Quality Guarantee

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Key Properties

No computed properties available.

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Protocol Information

PNU-282987 (orb1305505)

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% DMSO +
%+
% Tween 80 +
%

Available Sizes

Select a size below

5 mg
$ 80.00
10 mg
$ 110.00
1 ml x 10 mM (in DMSO)
$ 120.00
25 mg
$ 180.00
50 mg
$ 280.00
100 mg
$ 380.00
200 mg
$ 540.00
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