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PF 429242

PF 429242

Catalog Number: orb1302957

DispatchUsually dispatched within 3-5 working days
$ 140.00
Catalog Numberorb1302957
CategorySmall Molecules
DescriptionPF 429242
Purity99.27%
MW409.56
Biological ActivityPF-429242 is a competitive inhibitor of sterol regulatory element-binding protein (SREBP) site 1 protease (IC50 = 0.175 μM). It is selective for site 1 protease against a panel of serine proteases. PF-429242 inhibits rate of cholesterol synthesis in CHO cells (IC50 = 0.53 μM).
CAS Number[947303-87-9]
FormulaC25H35N3O2
SMILESN(C(=O)C1=CC=C(CN(CC)CC)C=C1)(CCC2=C(OC)C=CC=C2)[C@@H]3CCNC3
Storage-20°C
NoteFor research use only
  • PF 429242 [orb1222973]

    > 98% (HPLC)

    947303-87-9

    482.5

    C25H35N3O2·2HCl

    1 g, 500 mg, 200 mg, 100 mg, 2 mg, 5 mg, 10 mg, 25 mg, 50 mg