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GRK2 Inhibitor 2

SKU: orb2277567

Description

This potent small molecule inhibitor targets GRK2 (IC50 = 19 nM) and Aurora A kinase. It is used in cardiovascular research, particularly for studying congestive heart failure mechanisms, as it enhances β-adrenergic receptor signaling and cAMP production in cellular models.

Research Area

Cell Biology, Epigenetics & Chromatin, Pharmacology & Drug Discovery

Images & Validation

Key Properties

CAS Number2592436-21-8
MW332.36
FormulaC19H16N4O2
SMILESO=C1C=2C(=CC=C(C2)C=3C=NNC3)C=NN1CC4=CC(OC)=CC=C4
TargetAurora Kinase,GRK,Others

Storage & Handling

Storage-20°C
Expiration Date12 months from date of receipt.
DisclaimerFor research use only

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Quality Guarantee

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Key Properties

No computed properties available.

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GRK2 Inhibitor 2 (orb2277567)

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