GSK466317A

SKU: orb1700458

Description

GSK466317A is a potent and selective small molecule inhibitor of G protein-coupled receptor kinase 2 (GRK2). This compound is a valuable research tool for investigating GRK2's role in cellular signaling, heart failure, and metabolic studies in both in vitro and in vivo experimental models.

Research Area

Pharmacology & Drug Discovery, Signal Transduction

Key Properties

• CAS Number: 864082-48-4
• MW: 448.83
• Formula: C₂₁H₁₆ClF₃N₄O₂
• SMILES: C(NC=1C=C2C(=C(Cl)C1)NN=C2)(=O)C=3C(CC(=O)NC3C)C4=CC=C(C(F)(F)F)C=C4
• Target: PKA,GRK,Others

Storage & Handling

• Storage: -20°C
• Expiration Date: 12 months from date of receipt.
• Disclaimer: For research use only

Compound Identifiers

PubChem CID

11751266