CMPD101

Catalog Number: orb1308435

Catalog Number	orb1308435
Category	Small Molecules
Description	CMPD101
CAS Number	865608-11-3
Purity	99.01%
MW	466.46
SMILES	Cn1c(CNc2cccc(c2)C(=O)NCc2ccccc2C(F)(F)F)nnc1-c1ccncc1
Formula	C₂₄H₂₁F₃N₆O
Biological Activity	CMPD101 is a membrane-permeable small-molecule inhibitor of GRK2/3 (IC50: 18 nM and 5.4 nM). Which can be used for the study of heart failure. CMPD101 exhibits less selectively against GRK1, GRK5, ROCK-2 and PKCα with IC50s of 3.1 μM , 2.3 μM, 1.4 μM and 8.1 μM, respectively.
Storage	-20°C
Note	For research use only
Expiration Date	12 months from date of receipt.

CMPD101 hydrochloride [orb2664173]
Purity:
98.00%
CAS Number:
1941168-71-3
MW:
502.92
Formula:
C₂₄H₂₂ClF₃N₆O
Sizes Available: 50 mg, 10 mg
Compound 101 [orb2655617]
Purity:
> 98% (HPLC)
CAS Number:
865608-11-3
MW:
466.5
Formula:
C₂₄H₂₁F₃N₆O
Sizes Available: 5 mg, 10 mg, 25 mg, 50 mg
Compound 101 [orb746258]
CAS Number:
[865608-11-3]
Sizes Available: 1 ml x 10 mm (in DMSO), 1 g, 100 mg, 250 mg