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ERK1/2 inhibitor 8

SKU: orb1686712

Description

ERK1/2 inhibitor 8 is a highly potent and selective small molecule targeting ERK2 with an IC50 of 0.48 nM. It is a valuable research tool for investigating the MAPK/ERK pathway in cancer and other diseases, enabling both in vitro cellular studies and in vivo preclinical research.

Research Area

Pharmacology & Drug Discovery; Cell Biology

Images & Validation

Key Properties

CAS Number2648368-43-6
MW493.97
FormulaC23H20ClN7O2S
SMILESC(N1C2(C3=C(C1=O)N=C(S3)C4=NC(NC=5N(C)N=CC5)=NC=C4C)COC2)C6=CC(Cl)=CC=C6
TargetERK,Others

Storage & Handling

Storage-20°C
Expiration Date12 months from date of receipt.
DisclaimerFor research use only

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Key Properties

No computed properties available.

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Protocol Information

ERK1/2 inhibitor 8 (orb1686712)

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