Cart summary

You have no items in your shopping cart.

Endoxifen

Endoxifen

Catalog Number: orb1302991

DispatchUsually dispatched within 3-5 working days
$ 150.00
Catalog Numberorb1302991
CategorySmall Molecules
DescriptionEndoxifen
Purity99.66%
MW373.49
Biological Activity(E/Z)-Endoxifen ((E/Z)-Endoxifen) is an active metabolite of tamoxifen produced by the sequential action of cytochrome P450 (CYP) isoforms, including CYP2D6. It is a strong anti-estrogen, as it has an approximately 100-fold greater affinity for estrogen receptors than tamoxifen. As the efficient conversion of tamoxifen to endoxifen depends on CYP2D6, polymorphisms in this CYP isoform can impact the effectiveness of TMX treatment.
CAS Number110025-28-0
FormulaC25H27NO2
SMILESCC\C(=C(\c1ccc(O)cc1)c1ccc(OCCNC)cc1)c1ccccc1
Storage-20°C
NoteFor research use only
  • EGFR-IN-43 [orb1982922]

    98.00%

    860.45

    C50H55ClFN5O5

    50 mg, 5 mg
  • EGFR-IN-42 [orb1982923]

    98.00%

    846.43

    C49H53ClFN5O5

    50 mg, 5 mg
  • Endoxifen mesylate [orb1737902]

    98.00%

    1032008-71-1

    469.59

    C26H31NO5S

    25 mg, 100 mg, 50 mg
  • Endoxifen E-isomer hydrochloride [orb1693727]

    96.47%

    [1197194-61-8]

    409.95

    C25H28ClNO2

    5 mg, 1 mg, 1 ml x 10 mM (in DMSO)
  • Endoxifen Z-isomer hydrochloride [orb1685547]

    98.00%

    [1032008-74-4]

    409.95

    C25H28ClNO2

    2 mg