You have no items in your shopping cart.
Cart summary
Endoxifen mesylate
Catalog Number: orb1737902
| Catalog Number | orb1737902 |
|---|---|
| Category | Small Molecules |
| Description | Endoxifen mesylate |
| CAS Number | 1032008-71-1 |
| Purity | 0.98 |
| MW | 469.59 |
| SMILES | S(C)(=O)(=O)O.C(=C(/CC)\C1=CC=CC=C1)(\C2=CC=C(OCCNC)C=C2)/C3=CC=C(O)C=C3 |
| Formula | C26H31NO5S |
| Biological Activity | Endoxifen, also known as N-desmethyl-4-hydroxytamoxifen, is a chemical that is under development for estrogen receptor-positive breast cancer. It is also being evaluated as an antipsychotic for treatment of mania and other psychotic disorders. Endoxifen is a nonsteroidal selective estrogen receptor modulator (SERM) of the triphenylethylene group. It is an active metabolite of tamoxifen and has been found to be effective in patients that have failed previous hormonal therapies (tamoxifen, aromatase inhibitors, and fulvestrant). The prodrug tamoxifen is metabolized by the CYP2D6 enzyme to produce afimoxifene (4-hydroxytamoxifen) and endoxifen. |
| Storage | -20°C |
| Note | For research use only |
| Expiration Date | 12 months from date of receipt. |
