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CBP-IN-1

SKU: orb1944321

Description

CBP-IN-1 is a potent and selective CBP inhibitor with an IC50 of 1.5 nM, also inhibiting CBP BRET and BRD4(1) at higher concentrations. This small molecule is a valuable chemical probe for epigenetic research, enabling the study of CBP/p300 function in cancer models and transcriptional regulation in both cellular and biochemical assays.

Research Area

Epigenetics & Chromatin

Images & Validation

Key Properties

CAS Number1936431-44-5
MW509.59
FormulaC27H33F2N7O
SMILESC(C)(=O)N1CC=2C(=NN(C2CC1)C3CCNCC3)N4C=5C(=CC(=C(C(F)F)C5)C6=CN(C)N=C6)CCC4
TargetEpigenetic Reader Domain

Storage & Handling

Storage-20°C
Expiration Date12 months from date of receipt.
DisclaimerFor research use only

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Quality Guarantee

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Key Properties

No computed properties available.

Protocol Information