Queen's Award Received in 2021 ISO 9001 Certified Delivered over 1,000,000 bio-reagents to life science researchers Trusted by Life Science Communities
Cart summary

You have no items in your shopping cart.

CBP-IN-1

SKU: orb1944321

Description

CBP-IN-1 is a potent and selective CBP inhibitor with an IC50 of 1.5 nM, also inhibiting CBP BRET and BRD4(1) at higher concentrations. This small molecule is a valuable chemical probe for epigenetic research, enabling the study of CBP/p300 function in cancer models and transcriptional regulation in both cellular and biochemical assays.

Research Area

Epigenetics & Chromatin

Images & Validation

Key Properties

CAS Number1936431-44-5
MW509.59
FormulaC27H33F2N7O
SMILESC(C)(=O)N1CC=2C(=NN(C2CC1)C3CCNCC3)N4C=5C(=CC(=C(C(F)F)C5)C6=CN(C)N=C6)CCC4
TargetEpigenetic Reader Domain

Storage & Handling

Storage-20°C
Expiration Date12 months from date of receipt.
DisclaimerFor research use only

Similar Products

  • Inobrodib [orb1309860]

    99.18% (May vary between batches)

    2222941-37-7

    534.6

    C30H32F2N4O3

    100 mg, 1 mg, 2 mg, 1 ml x 10 mM (in DMSO), 5 mg, 10 mg, 25 mg, 50 mg
  • β-catenin/CBP-IN-1 [orb1708814]

    1198780-38-9

    658.64

    C33H35N6O7P

    25 mg
  • CBP-IN-1 [orb1219374]

    >98% (HPLC)

    2222941-37-7

    534.6

    C30H32F2N4O3

    5 mg, 50 mg, 200 mg, 25 mg, 1 g, 500 mg, 2 mg, 100 mg, 10 mg
Quality Guarantee

Quality Guarantee

Explore bioreagents carefree to elevate your research. All our products are rigorously tested for performance. If a product does not perform as described on its datasheet, our scientific support team will provide expert troubleshooting, a prompt replacement, or a refund. For full details, please see our Terms & Conditions and Buying Guide. Contact us at [email protected].

Key Properties

No computed properties available.

Documents Download

Datasheet
Product Information
Download

Request a Document

Protocol Information

CBP-IN-1 (orb1944321)

  • Star
  • Star
  • Star
  • Star
  • Star
  • 0.0
Based on 0 reviews

Participating in our Biorbyt product reviews program enables you to support fellow scientists by sharing your firsthand experience with our products.

Login to Submit a Review

No reviews yet

Step 1: Enter information below

(Recommended: An additional animal making an allowance for loss during the experiment)

Step 2: Enter the in vivo formulation

(This is only the calculator, not formulation. Please contact us first if there is no in vivo formulation at the solubility Section.)

% DMSO +
%+
% Tween 80 +
%