Inobrodib

SKU: orb1309860

Description

Inobrodib (CBP-IN-1) is a potent and selective small molecule inhibitor targeting the bromodomain of the p300/CBP proteins. This compound is a valuable chemical probe for epigenetic research, enabling the study of transcriptional regulation and oncogenesis in both cellular and animal models.

Research Area

Epigenetics & Chromatin

Key Properties

• CAS Number: 2222941-37-7
• MW: 534.6
• Purity: 99.18% (May vary between batches)
• Formula: C₃₀H₃₂F₂N₄O₃
• SMILES: CO[C@H]1CC[C@@H](CC1)n1c(nc2cc(ccc12)-c1c(C)noc1C)[C@@H]1CCCC(=O)N1c1ccc(F)c(F)c1
• Target: Epigenetic Reader Domain
• Solubility: 10% DMSO+40% PEG300+5% Tween 80+45% Saline:5 mg/mL (9.35 mM);DMSO:100 mg/mL (187.06 mM)

Storage & Handling

• Storage: keep away from moisture,store at low temperature | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature.
• Expiration Date: 12 months from date of receipt.
• Disclaimer: For research use only

Alternative Names

CBP-IN-1, CCS 1477, CCS1477, CCS-1477, bromodomain, cancer, Epigenetic Reader Domain, EpigeneticReaderDomain, Inobrodib, Inhibitor, histones, inhibit, oral, nude, mice, p300/CBP, prostate, proliferation

Compound Identifiers

PubChem CID

134457551