AR antagonist 9

SKU: orb2814450

Description

AR antagonist 9 is a potent, orally bioavailable androgen receptor (AR) antagonist that disrupts AR dimerization. It exhibits activity comparable to Enzalutamide against wild-type AR and shows superior efficacy against common resistance mutants like ARF876L/T877A. This compound demonstrates significant oral bioavailability and inhibits tumor growth in LNCaP xenograft models, supporting its research in overcoming prostate cancer resistance.

Research Area

Metabolism Research, Pharmacology & Drug Discovery

Images & Validation

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Key Properties

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MW	351.29
Formula	C₁₈H₁₃F₄NO₂
Target	Androgen Receptor

Storage & Handling

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Storage	-20°C
Expiration Date	12 months from date of receipt.
Disclaimer	For research use only

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Gene Symbol

Androgen Receptor

Protocol Information

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Purity:	0.98
CAS Number:	13523-86-9
MW:	248.32
Formula:	C₁₄H₂₀N₂O₂

CAS Number:	1431166-12-9
MW:	294.27
Formula:	C₁₅H₁₃F₃N₂O

CAS Number:	2412715-30-9
MW:	368.55
Formula:	C₂₅H₃₆O₂

CAS Number:	1790308-86-9
MW:	346.44
Formula:	C₁₈H₂₂N₂O₃S

Purity:	99.07% (May vary between batches)
CAS Number:	1818885-54-9
MW:	278.777
Formula:	C₁₅H₁₉ClN₂O

AR antagonist 9

Description

Research Area

Images & Validation

Key Properties

Storage & Handling

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