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Adenosine receptor inhibitor 1

SKU: orb1688187

Description

Adenosine receptor inhibitor 1 is a potent and selective pan-AR antagonist with high affinity for the A2A subtype (Ki = 68.5 nM). It demonstrates antinociceptive and anti-inflammatory activities in vivo, making it a valuable research tool for studying cancer, neuroinflammation, and neurodegenerative diseases.

Research Area

Neuroscience, Pharmacology & Drug Discovery

Images & Validation

Key Properties

CAS Number2550400-52-5
MW395.82
FormulaC17H19ClFN5O3
SMILESCN1C2=C(N(C)C(NCC3=C(F)C(OC)=CC=C3Cl)=N2)C(=O)N(CC)C1=O
TargetAdenosine Receptor,Others

Storage & Handling

Storage-20°C
Expiration Date12 months from date of receipt.
DisclaimerFor research use only

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Key Properties

No computed properties available.

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Protocol Information

Adenosine receptor inhibitor 1 (orb1688187)

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