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ZEN-2759

SKU: orb2900589

Description

ZEN-2759 is a potent BET (Bromodomain and Extra-Terminal Domain) inhibitor, with IC50 values of 0.23, 0.08 and 0.28 μM for BRD4(BD1), BRD4(BD2), and BRD4(BD1BD2), respectively.

Images & Validation

Key Properties

CAS Number1616400-50-0
MW280.32
Purity>98% (HPLC)
FormulaC17H16N2O2
SMILESCC=1C(C2=CN(CC3=CC=CC=C3)C(=O)C=C2)=C(C)ON1
TargetEpigenetic Reader Domain
SolubilityIn Vitro: DMSO : 100 mg/mL (356.74 mM; Ultrasonic )

Storage & Handling

StorageStorage temperature: -20°C. Stability: ≥ 2 years
Expiration Date12 months from date of receipt.
DisclaimerFor research use only

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Protocol Information

ZEN-2759 (orb2900589)

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% DMSO +
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Available Sizes

Select a size below

2 mg
$ 140.00
5 mg
$ 180.00
10 mg
$ 260.00
25 mg
$ 400.00
50 mg
$ 590.00
100 mg
$ 790.00
500 mg
$ 1,620.00