TRPM4 inhibitor 8

SKU: orb1685221

Description

TRPM4 inhibitor 8 is a small molecule compound that selectively blocks the Transient Receptor Potential Melastatin 4 (TRPM4) channel. Its application in research includes studying TRPM4's role in cellular processes like proliferation and migration, both in vitro and in vivo, particularly in models of cancer, cardiovascular, and immune-related diseases.

Research Area

Neuroscience, Pharmacology & Drug Discovery, Pharmacology & Drug Discovery; Cell Biology, Signal Transduction

Key Properties

• CAS Number: 1353979-43-7
• MW: 257.17
• Purity: 99.84% (May vary between batches)
• Formula: C₁₁H₁₇BrN₂
• SMILES: CCN(CCN)Cc1cccc(Br)c1
• Target: TRP/TRPV Channel,iGluR,ERK
• Solubility: DMSO:70 mg/mL (272.19 mM)

Storage & Handling

• Storage: -20°C
• Expiration Date: 12 months from date of receipt.
• Disclaimer: For research use only

Alternative Names

brain damage, iGluR, hippocampal neurons, Inhibitor, Extracellular signal regulated kinases, ERK, inhibit, Ionotropic glutamate receptors, neurodegenerative diseases, neuroprotective activity, TRP Channel, Transient receptor potential channels, transient receptor potential cation channel subfamily M member 4, TRPVChannel, TRPV Channel, TRPM4, TRPM4 inhibitor 8, TRPM-4 inhibitor 8, TRPChannel

Compound Identifiers

PubChem CID

66568274