Trimebutine maleate

SKU: orb1309442

Description

Trimebutine maleate is a spasmolytic agent that acts as a weak agonist at mu-opioid receptors and exhibits antimuscarinic activity. It is utilized in research on gastrointestinal motility disorders, with applications in both in vitro receptor binding studies and in vivo models of abdominal pain.

Research Area

Cell Biology, Immunology & Inflammation, Metabolism Research, Neuroscience, Pharmacology & Drug Discovery, Signal Transduction

Key Properties

• CAS Number: 34140-59-5
• MW: 503.55
• Purity: 99.98% (May vary between batches)
• Formula: C₂₆H₃₃NO₉
• SMILES: OC(=O)/C=C\C(=O)O.CCC(COC(=O)c1cc(OC)c(OC)c(OC)c1)(N(C)C)c1ccccc1
• Target: Opioid Receptor,JNK,Akt,IRAK,Calcium Channel,ERK,NF-κB,Apoptosis,TLR,OCT,Potassium Channel
• Solubility: DMSO:55 mg/mL (109.22 mM);10% DMSO+40% PEG300+5% Tween 80+45% Saline:2 mg/mL (3.97 mM)

Storage & Handling

• Storage: Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature.
• Expiration Date: 12 months from date of receipt.
• Disclaimer: For research use only

Alternative Names

CalciumChannel, Calcium Channel, Inhibitor, Debridat, OpioidReceptor, Opioid Receptor, inhibit, Polibutin, Trimebutine, Trimebutine maleate, Trimebutine Maleate

Compound Identifiers

PubChem CID

5388977