TNKS1/2-IN-1

SKU: orb1744566

Description

TNKS1/2-IN-1 is a potent, cell-active tankyrase (TNKS1/2) inhibitor with pIC50 values of 7.1-8.2. It is widely used in biochemical and cellular research to study the roles of tankyrases in cancer, fibrosis, and hyperproliferative diseases, including in vitro Wnt/β-catenin pathway modulation.

Research Area

Epigenetics & Chromatin, Molecular Biology, Signal Transduction

Key Properties

• CAS Number: 1498300-31-4
• MW: 517.47
• Formula: C₂₆H₂₃F₄N₃O₄
• SMILES: C(N1C=2C(C(=O)N(C[C@@H]3CC[C@@H](C(O)=O)CC3)C1=O)=C(C)C(F)=CC2)C4=C(C#N)C(C(F)(F)F)=CC=C4
• Target: PARP,Others

Storage & Handling

• Storage: -20°C
• Expiration Date: 12 months from date of receipt.
• Disclaimer: For research use only

Compound Identifiers

PubChem CID

72549541