Cart summary

You have no items in your shopping cart.

SB 242084

SKU: orb1299955

Description

SB 242084 is a selective 5-HT2C receptor antagonist used as a research chemical. It is applied in neuroscience studies to investigate receptor function in models of depression, anxiety, and feeding behavior, utilizing both in vitro and in vivo experimental systems.

Research Area

Neuroscience, Pharmacology & Drug Discovery

Images & Validation

Key Properties

CAS Number181632-25-7
MW394.85
Purity98.00%
FormulaC21H19ClN4O2
SMILESCc1cc2CCN(C(=O)Nc3ccc(Oc4cccnc4C)nc3)c2cc1Cl
Target5-HT Receptor
SolubilityDMSO:44 mg/mL (111.43 mM);10% DMSO+40% PEG300+5% Tween 80+45% Saline:2 mg/mL (5.07 mM)

Bioactivity

Target IC50
5 hT2C receptor:9.0 (pKi)

Storage & Handling

StoragePowder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature.
DisclaimerFor research use only

Alternative Names

5HTReceptor, 5-HT Receptor, 5-HT2C, 5HT Receptor, SB 242084, SB242084, SB-242084

Similar Products

  • SB 242084 monohydrochloride [orb2664011]

    1260505-34-7

    431.32

    C21H20Cl2N4O2

    50 mg, 10 mg
  • SB 242084 dihydrochloride [orb1693152]

    1049747-87-6

    467.78

    C21H21Cl3N4O2

    2 mg
  • SB 242084 [orb1225878]

    >98% (HPLC)

    181632-25-7

    467.8

    C21H19ClN4O2

    100 mg, 2 mg, 5 mg, 25 mg, 50 mg, 10 mg, 1 g, 500 mg, 200 mg
Quality Guarantee

Quality Guarantee

Explore bioreagents carefree to elevate your research. All our products are rigorously tested for performance. If a product does not perform as described on its datasheet, our scientific support team will provide expert troubleshooting, a prompt replacement, or a refund. For full details, please see our Terms & Conditions and Buying Guide. Contact us at [email protected].

Key Properties

No computed properties available.

Documents Download

Datasheet
Product Information
Download

Request a Document

Protocol Information

SB 242084 (orb1299955)

  • Star
  • Star
  • Star
  • Star
  • Star
  • 0.0
Based on 0 reviews

Participating in our Biorbyt product reviews program enables you to support fellow scientists by sharing your firsthand experience with our products.

Login to Submit a Review

No reviews yet

Step 1: Enter information below

(Recommended: An additional animal making an allowance for loss during the experiment)

Step 2: Enter the in vivo formulation

(This is only the calculator, not formulation. Please contact us first if there is no in vivo formulation at the solubility Section.)

% DMSO +
%+
% Tween 80 +
%

Available Sizes

Select a size below

1 mg
$ 80.00
5 mg
$ 130.00
1 ml x 10 mM (in DMSO)
$ 140.00
10 mg
$ 160.00
25 mg
$ 300.00
50 mg
$ 470.00
100 mg
$ 700.00
DispatchUsually dispatched within 3-5 working days
Bulk Enquiry