SB 242084 dihydrochloride

SKU: orb1693152

Description

SB 242084 hydrochloride is a potent and selective 5-HT2C receptor antagonist with a pKi of 9.0, exhibiting 158-fold and 100-fold selectivity over 5-HT2A and 5-HT2B receptors, respectively. This compound is a valuable pharmacological tool used in vitro and in vivo to investigate the role of 5-HT2C receptors in anxiety, depression, and feeding behavior.

Research Area

Neuroscience, Pharmacology & Drug Discovery

Images & Validation

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Key Properties

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CAS Number	1049747-87-6
MW	467.78
Formula	C₂₁H₂₁Cl₃N₄O₂
SMILES	Cl.Cl.Cc1cc2CCN(C(=O)Nc3ccc(Oc4cccnc4C)nc3)c2cc1Cl
Target	Others,5-HT Receptor

Storage & Handling

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Storage	-20°C
Expiration Date	12 months from date of receipt.
Disclaimer	For research use only

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Compound Identifiers

PubChem CID

16219981 ↗

Key Properties

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No computed properties available.

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