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(R)-Elagolix

SKU: orb1309714

Description

(R)-Elagolix

Research Area

Pharmacology & Drug Discovery

Images & Validation

Key Properties

CAS Number834153-87-6
MW631.59
Purity99.08%
FormulaC32H30F5N3O5
SMILES[H][C@@](Cn1c(=O)c(c(C)n(Cc2c(F)cccc2C(F)(F)F)c1=O)-c1cccc(OC)c1F)(NCCCC(O)=O)c1ccccc1
TargetGNRH Receptor
Solubility10% DMSO+40% PEG300+5% Tween 80+45% Saline:4 mg/mL (6.33 mM);DMSO:100 mg/mL (158.33 mM)

Bioactivity

Target IC50
NFAT:5.4 nM|GnRHR:0.25 nM|GnRHR:3.7 nM (Ki)

Storage & Handling

Storagestore at low temperature | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature.
DisclaimerFor research use only

Alternative Names

Elagolix, Gonadotropin releasing hormone receptor, GNRHReceptor, GNRHR, GnRHR, GnRH Receptor, GNRH Receptor, inhibit, Inhibitor, NBI 56418, NBI56418, NBI-56418, (R) Elagolix, (R)Elagolix, (R)-Elagolix

Similar Products

  • (R)-Elagolix [orb1217613]

    >98% (HPLC)

    834153-87-6

    631.6

    C32H30F5N3O5

    1 g, 500 mg, 25 mg, 200 mg, 5 mg, 10 mg, 2 mg, 50 mg, 100 mg
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Key Properties

No computed properties available.

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(R)-Elagolix (orb1309714)

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% DMSO +
%+
% Tween 80 +
%

Available Sizes

Select a size below

5 mg
$ 90.00
1 ml x 10 mM (in DMSO)
$ 110.00
10 mg
$ 120.00
25 mg
$ 190.00
50 mg
$ 260.00
100 mg
$ 390.00
200 mg
$ 550.00
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