(R)-Elagolix

• Catalog Number: orb1309714
• Category: Small Molecules
• Description: (R)-Elagolix
• CAS Number: 834153-87-6
• Purity: 97.63%
• MW: 631.59
• SMILES: CC1=C(C(=O)N(C[C@H](NCCCC(O)=O)C2=CC=CC=C2)C(=O)N1CC3=C(C(F)(F)F)C=CC=C3F)C4=C(F)C(OC)=CC=C4
• Formula: C₃₂H₃₀F₅N₃O₅
• Biological Activity: (R)-Elagolix (NBI-56418) is a short-acting, nonpeptide, GnRH antagonist with an IC50 and Ki of 0.25 and 3.7 nM, respectively. administered orally, that unlike injectable depot GnRH agonists and antagonists, produces a dose-dependent suppression of ovarian estrogen production, that is, from partial suppression at lower doses to full suppression at higher doses.
• Note: For research use only
• Expiration Date: 12 months from date of receipt.