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MRK-016

SKU: orb611735

Description

A potent, functionally selective, CNS-penetrating and orally bioavailable inverse agonist of benzodiazepine site of GABAA α5 receptor with Ki of 0.8-1.5 nM for α1-, α2-, α3-, andα5-containing GABAA receptors.

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Key Properties

CAS Number342652-67-9
MW368.3931
FormulaC17H20N8O2
SMILESCN1C(COC2C(C(C)(C)C)=C3N(C(=NN=C3)C3C=C(C)ON=3)N=2)=NC=N1

Storage & Handling

DisclaimerFor research use only

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  • MRK-016 [orb2893738]

    99.76%

    342652-67-9

    368.39

    C17H20N8O2

    1 ml x 10 mM (in DMSO), 5 mg, 10 mg, 25 mg, 50 mg, 1 mg
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Protocol Information

MRK-016 (orb611735)

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10 mg
$ 220.00
50 mg
$ 840.00
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