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GPR40 agonist 7

SKU: orb2566163

Description

Compound 1 (GPR40 agonist 7) is an orally bioavailable small molecule agonist of GPR40. It stimulates insulin and GLP-1 secretion, demonstrating in vivo hypoglycemic activity with an ED50 of 0.58 mg/kg, making it a useful research tool for studying diabetes and metabolic disorders.

Research Area

Metabolism Research, Pharmacology & Drug Discovery

Images & Validation

Key Properties

CAS Number1821647-46-4
MW562.1
FormulaC29H40ClN3O6
SMILESC(C(O)=O)[C@@H]1N(C[C@H](OCCCOC)[C@H]1C)C2=CC=C(O[C@H]3[C@H](C)CN(CC3)C=4C=C(OC)N=CC4Cl)C=C2
TargetGPCR

Storage & Handling

Storage-20°C
Expiration Date12 months from date of receipt.
DisclaimerFor research use only

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Key Properties

No computed properties available.

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Protocol Information

GPR40 agonist 7 (orb2566163)

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Step 1: Enter information below

(Recommended: An additional animal making an allowance for loss during the experiment)

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