CMPD101 hydrochloride

SKU: orb2664173

Description

CMPD101 hydrochloride is a potent, cell-permeable inhibitor of GRK2 (IC50=18 nM) and GRK3 (IC50=5.4 nM), with additional activity against ROCK-2 and PKCα. This tool compound is utilized in cardiovascular and oncology research to investigate GPCR signaling pathways in both cellular and animal models.

Images & Validation

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Key Properties

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CAS Number	1941168-71-3
MW	502.92
Formula	C₂₄H₂₂ClF₃N₆O
SMILES	Cl.O=C(NCC=1C=CC=CC1C(F)(F)F)C=2C=CC=C(C2)NCC3=NN=C(C=4C=CN=CC4)N3C

Storage & Handling

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Storage	-20°C
Expiration Date	12 months from date of receipt.
Disclaimer	For research use only

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Compound Identifiers

PubChem CID

137797638 ↗

Key Properties

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No computed properties available.

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