CMPD101 hydrochloride

• Catalog Number: orb2664173
• Category: Small Molecules
• Description: CMPD101 hydrochloride is a membrane-permeable small molecule inhibitor of GRK2 and GRK3, exhibiting IC50 values of 18 nM and 5.4 nM, respectively. This compound also inhibits Rho-associated kinase 2 (ROCK-2) and PKCα, with IC50 values of 1.4 μM and 8.1 μM, respectively.
• CAS Number: 1941168-71-3
• Purity: 98.00%
• MW: 502.92
• SMILES: Cl.O=C(NCC=1C=CC=CC1C(F)(F)F)C=2C=CC=C(C2)NCC3=NN=C(C=4C=CN=CC4)N3C
• Formula: C₂₄H₂₂ClF₃N₆O
• Storage: -20°C
• Note: For research use only
• Expiration Date: 12 months from date of receipt.