CMPD101 hydrochloride

SKU: orb2664173

Description

CMPD101 hydrochloride is a potent, cell-permeable inhibitor of GRK2 (IC50=18 nM) and GRK3 (IC50=5.4 nM), with additional activity against ROCK-2 and PKCα. This tool compound is utilized in cardiovascular and oncology research to investigate GPCR signaling pathways in both cellular and animal models.

Key Properties

• CAS Number: 1941168-71-3
• MW: 502.92
• Formula: C₂₄H₂₂ClF₃N₆O
• SMILES: Cl.O=C(NCC=1C=CC=CC1C(F)(F)F)C=2C=CC=C(C2)NCC3=NN=C(C=4C=CN=CC4)N3C

Storage & Handling

• Storage: -20°C
• Expiration Date: 12 months from date of receipt.
• Disclaimer: For research use only

Compound Identifiers

PubChem CID

137797638