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CK1-IN-1

SKU: orb1221006

Description

CK1-IN-1 compound 1c reported in patent WO2015119579A1 is a casein kinase 1 (CK1) inhibitor. It has IC50s of 15 nM 16 nM 73 nM for CK1δ and CK1ε p38σ MAPK respectively.

Images & Validation

Key Properties

CAS Number1784751-20-7
MW383.39
Purity>98% (HPLC)
FormulaC24H15F2N3
SMILESFc1ccc(cc1)-c1nc([nH]c1-c1ccncc1)-c1ccc2ccccc2c1F
TargetCasein Kinase
SolubilityDMSO: 60 mg/mL (156.5 mM); Water: Insoluble

Storage & Handling

StorageStorage temperature: -20°C. Stability: ≥ 2 years
Expiration Date12 months from date of receipt.
DisclaimerFor research use only

Alternative Names

PUN51207

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CK1-IN-1 (orb1221006)

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200 mg
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50 mg
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100 mg
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