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BI-4464

SKU: orb1220934

Description

BI-4464 is a highly selective ATP competitive inhibitor of PTK2/FAK with an IC50 of 17 nM. A PTK2 ligand for PROTAC.

Images & Validation

Key Properties

CAS Number1227948-02-8
MW555.56
Purity>98% (HPLC)
FormulaC28H28F3N5O4
SMILESCOc1cc(ccc1Nc1ncc(c(Oc2cccc3CCC(=O)c23)n1)C(F)(F)F)C(=O)NC1CCN(C)CC1
TargetFAK
SolubilityDMSO:16.67 mg/mL (30.01 mM)

Storage & Handling

StorageStorage temperature: -20°C. Stability: ≥ 2 years
Expiration Date12 months from date of receipt.
DisclaimerFor research use only

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Protocol Information

BI-4464 (orb1220934)

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% DMSO +
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% Tween 80 +
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Available Sizes

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200 mg
500 mg
2 mg
$ 150.00
5 mg
$ 250.00
10 mg
$ 390.00
25 mg
$ 620.00
50 mg
$ 920.00
100 mg
$ 1,330.00