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A-836339

SKU: orb1223516

Description

A-836339 (A836339) is a potent and selective cannabinoid CB2 receptor agonist with Ki of 0.64 and 0.76 nM for human and rat CB2 receptors, displays 425- and 189-fold selectivity over CB1 receptor, respectively; exhibits full agonist efficacy (Emax=102%) with high potency (EC50=1.6 nM), greater potency than other CB2-selective ligands including JWH-015 and GW-842166X; exhibits a potent CB2 receptor-mediated antihyperalgesic effect in various animal pain models, also demonstrates efficacies in the chronic constrain injury (CCI) model of neuropathic pain.

Images & Validation

Key Properties

CAS Number959746-77-1
MW310.4548
Purity>98% (HPLC)
FormulaC16H26N2O2S
SMILESCC1=C(C)N(CCOC)/C(S1)=N/C(C2C(C)(C)C2(C)C)=O
TargetCannabinoid Receptor
SolubilityDMSO: 12 mg/mL

Storage & Handling

StorageStorage temperature: -20°C. Stability: ≥ 2 years
Expiration Date12 months from date of receipt.
DisclaimerFor research use only

Alternative Names

A836339

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A-836339 (orb1223516)

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Available Sizes

Select a size below

200 mg
500 mg
5 mg
$ 230.00
10 mg
$ 390.00
25 mg
$ 630.00
50 mg
$ 910.00
100 mg
$ 1,280.00