YM-254890

SKU: orb1988853

Description

YM-254890 is a macrocyclic hexapeptide and a potent, selective inhibitor of Gαq/11 proteins. It effectively blocks ADP-induced platelet aggregation and Gq-mediated signaling pathways, making it a valuable tool for studying cardiovascular biology and GPCR mechanisms in both cellular and animal models.

Research Area

Neuroscience, Pharmacology & Drug Discovery

Key Properties

• CAS Number: 568580-02-9
• MW: 960.08
• Purity: 95.00%
• Formula: C₄₆H₆₉N₇O₁₅
• SMILES: CO[C@H](C)[C@@H]1N(C)C(=O)[C@@H](NC(=O)[C@H](C)N(C)C(=O)[C@H](C)NC(=O)C(=C)N(C)C(=O)[C@@H](Cc2ccccc2)OC(=O)[C@@H](NC(C)=O)[C@@H](C)OC1=O)[C@H](OC(=O)[C@@H](NC(C)=O)[C@H](O)C(C)C)C(C)C
• Target: P2Y Receptor

Storage & Handling

• Storage: -20°C
• Expiration Date: 12 months from date of receipt.
• Disclaimer: For research use only

Compound Identifiers

PubChem CID

9919454