YK-2-69

SKU: orb1739916

Description

YK-2-69 is a potent and selective small molecule inhibitor of DYRK2 kinase. It has demonstrated anti-proliferative effects in prostate cancer cell lines and has shown efficacy in reducing tumor growth in preclinical in vivo models, supporting its use as a research tool in oncology.

Research Area

Cell Biology, Signal Transduction

Key Properties

• CAS Number: 2619846-89-6
• MW: 506.6
• Purity: 99.92% (May vary between batches)
• Formula: C₂₅H₂₇FN₈OS
• SMILES: O=C(C1=CN=C(C=C1)NC=2N=CC(F)=C(N2)C=3C=CC=4N=C(SC4C3)N(C)C)N5CCN(CC)CC5
• Target: DYRK

Bioactivity

• Target IC50:
  DYRK2:9 nM

Storage & Handling

• Storage: -20°C
• Expiration Date: 12 months from date of receipt.
• Disclaimer: For research use only

Alternative Names

DYRK2

Compound Identifiers

PubChem CID

163183800