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WP1066
Catalog Number: orb1306297
| Catalog Number | orb1306297 |
|---|---|
| Category | Small Molecules |
| Description | WP1066 |
| CAS Number | 857064-38-1 |
| Purity | 99.73% |
| MW | 356.22 |
| SMILES | C(=C(/C(N[C@@H](C)C1=CC=CC=C1)=O)\C#N)\C=2N=C(Br)C=CC2 |
| Formula | C17H14BrN3O |
| Biological Activity | WP1066 is a inhibitor of JAK2 (IC50: 2.30 μM) and STAT3 (IC50: 2.43 μM) in HEL cells; shows activity to JAK2, STAT3/5, and ERK1/2, not JAK1 and JAK3. WP1066 has been used in trials studying the treatment of Melanoma, Brain Cancer, Solid Tumors, and Central Nervous System Neoplasms. |
| Note | For research use only |
| Expiration Date | 12 months from date of receipt. |
wp1066 (STAT Inhibitor III) [orb315333]
[857064-38-1]
356.2
C17H14BrN3O
100 mg, 250 mg, 1 g, 10 mM * 1 mL in DMSO
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