VU0238441

SKU: orb1299112

Description

VU0238441 is a selective agonist for the human muscarinic acetylcholine receptor M5, exhibiting an EC50 of 2.1 µM. This small molecule is a valuable research tool for investigating M5 receptor function in neuropharmacology, utilized in both in vitro assays and in vivo studies of central nervous system pathways.

Research Area

Neuroscience

Key Properties

• CAS Number: 85511-68-8
• MW: 339.7
• Purity: >99.99%
• Formula: C₁₆H₉ClF₃NO₂
• SMILES: FC(F)(F)c1ccc(CN2C(=O)C(=O)c3cccc(Cl)c23)cc1
• Target: AChR
• Solubility: DMSO:3.4 mg/mL (10.01 mM)

Bioactivity

• Target IC50:
  M5:2.1μM(EC50)

Storage & Handling

• Storage: Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature.
• Expiration Date: 12 months from date of receipt.
• Disclaimer: For research use only

Alternative Names

M5 mAChR, mAChR, Muscarinic acetylcholine receptor, inhibit, Inhibitor, VU 0238441, VU0238441, VU-0238441

Compound Identifiers

PubChem CID

44158142