VPC-13566

SKU: orb1304856

Description

VPC-13566 is a BF3 pocket-targeting small molecule that suppresses androgen receptor transcriptional activity by displacing the BAG1L peptide. It demonstrates efficacy in inhibiting the proliferation of prostate cancer cell lines in vitro and reducing the growth of AR-dependent xenograft tumors in vivo.

Research Area

Metabolism Research

Key Properties

• CAS Number: 218464-59-6
• MW: 258.32
• Purity: 99.55% (May vary between batches)
• Formula: C₁₈H₁₄N₂
• SMILES: CC1=C2C(C(=CN2)C3=NC4=C(C=C3)C=CC=C4)=CC=C1
• Target: Androgen Receptor
• Solubility: DMSO:65 mg/mL (251.63 mM)

Storage & Handling

• Storage: -20°C
• Expiration Date: 12 months from date of receipt.
• Disclaimer: For research use only

Alternative Names

Androgen Receptor, AndrogenReceptor, VPC 13566, VPC13566, VPC-13566

Compound Identifiers

PubChem CID

18729606