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Varenicline

Varenicline

Catalog Number: orb1690005

DispatchUsually dispatched within 8-10 weeks
$ 130.00
Catalog Numberorb1690005
CategorySmall Molecules
DescriptionVarenicline
Purity99.76%
MW211.26
Biological ActivityVarenicline (CP 526555), a cytisine-based nicotinic ligand, is a potent partial agonist for the α4β2 nicotinic acetylcholine receptor (nAChR) with an EC50 value of 2.3 μM and acts as a full agonist for α7 and α3β4 nAChRs, with respective EC50 values of 18 μM and 55 μM [1]. Notably, its effectiveness and potential in smoking cessation treatments are underscored by its pharmacological profile [2].
CAS Number[249296-44-4]
FormulaC13H13N3
SMILESN1=CC=NC2=CC3=C(C=C12)C4CNCC3C4
Storage-20°C
NoteFor research use only
  • Varenicline Tartrate [orb1225165]

    > 98%(HPLC)

    375815-87-5

    361.4

    C13H13N3·C4H6O6

    50 mg, 5 mg, 10 mg, 25 mg, 2 mg, 100 mg, 500 mg, 1 g
  • Varenicline [orb1221714]

    > 98% (HPLC)

    866823-63-4

    284.2

    C13H15Cl2N3

    200 mg, 5 mg, 10 mg, 25 mg, 50 mg, 100 mg, 1 g, 500 mg
  • Varenicline Hydrochloride [orb1703942]

    98.00%

    [230615-23-3]

    247.72

    C13H14ClN3

    5 mg, 2 mg, 1 ml x 10 mM (in DMSO)
  • Varenicline dihydrochloride [orb1303027]

    99.21%

    866823-63-4

    284.18

    C13H15Cl2N3

    10 mg, 50 mg, 100 mg, 5 mg, 25 mg, 1 ml x 10 mM (in DMSO)
  • Varenicline Tartrate [orb1307855]

    99.90%

    [375815-87-5]

    361.35

    C13H13N3·C4H6O6

    25 mg, 10 mg, 5 mg, 100 mg, 50 mg, 1 ml x 10 mM (in DMSO)