VA4 TG2 inhibitor

SKU: orb1739547

Description

VA4 is a novel, irreversible inhibitor that specifically targets the transamidase site of tissue transglutaminase (TG2). It is a valuable research tool for studying TG2's role in fibrotic diseases, celiac disease, and cancer in both cellular and animal models.

Research Area

Pharmacology & Drug Discovery, Protein Biochemistry

Key Properties

• CAS Number: 2088001-23-2
• MW: 635.77
• Formula: C₃₃H₄₁N₅O₆S
• SMILES: S(=O)(=O)(C=1C2=C(C(N(C)C)=CC=C2)C=CC1)N3CCN(C([C@@H](NC(OCC4=CC=CC=C4)=O)CCCCNC(C=C)=O)=O)CC3
• Target: Others,Glutaminase

Storage & Handling

• Storage: -20°C
• Expiration Date: 12 months from date of receipt.
• Disclaimer: For research use only

Compound Identifiers

PubChem CID

132024504