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Uprosertib

SKU: orb1223448

Description

Uprosertib (GSK2141795) is a selective, ATP-competitive, and orally bioavailable Akt inhibitor with IC50 of 180 nM, 328 nM, and 38 nM for Akt 1, 2 and 3, respectively. Phase 2.

Images & Validation

Key Properties

CAS Number1047634-65-0
MW429.3
Purity>98% (HPLC)
FormulaC18H16Cl2F2N4O2
TargetAkt1| Akt2| Akt3

Storage & Handling

StorageStorage temperature: -20°C. Stability: ≥ 2 years
Expiration Date12 months from date of receipt.
DisclaimerFor research use only

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Uprosertib (orb1223448)

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Available Sizes

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200 mg
500 mg
2 mg
$ 100.00
5 mg
$ 130.00
10 mg
$ 190.00
25 mg
$ 300.00
50 mg
$ 470.00
100 mg
$ 750.00