TRPV4 antagonist 3

SKU: orb1690682

Description

TRPV4 antagonist 3 is a potent and selective small molecule inhibitor of the TRPV4 ion channel, exhibiting an IC50 of 4.0 nM (pIC50 = 8.4). This compound is a valuable research tool for investigating TRPV4-mediated physiological and pathological processes in both cellular and animal models of pain, inflammation, and osmoregulation.

Research Area

Pharmacology & Drug Discovery, Pharmacology & Drug Discovery; Cell Biology

Images & Validation

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Key Properties

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CAS Number	2681273-35-6
MW	470.44
Formula	C₂₀H₁₈F₄N₄O₃S
SMILES	C[C@](N)(CCNS(=O)(=O)c1ccc(cc1C(F)(F)F)C#N)COc1ccc(C#N)c(F)c1
Target	TRP/TRPV Channel,Others

Storage & Handling

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Storage	-20°C
Expiration Date	12 months from date of receipt.
Disclaimer	For research use only

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Compound Identifiers

PubChem CID

162641390 ↗

Key Properties

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No computed properties available.

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