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TRPV1 antagonist 6

SKU: orb3133809

Description

TRPV1 antagonist 6 (compound 51) is a modality-selective TRPV1 antagonist that exhibits antagonistic activity against capsaicin activation with an IC50 of 2.85 nM and demonstrates an inhibition rate of 28.48% against proton activation at a concentration of 3 µM.

Images & Validation

Key Properties

FormulaC26H28ClN5O3
TargetTRP/TRPV Channel

Storage & Handling

Storage-20°C
Expiration Date12 months from date of receipt.
DisclaimerFor research use only

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TRPV1 antagonist 6 (orb3133809)

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