TRPV1 antagonist 10

SKU: orb3028095

Description

TRPV1 antagonist 10 is a potent, orally active TRPV1 antagonist with an IC50 of 33.06 nM and serves as a moderate to weak inhibitor of URAT1 (IC50 = 22.51 μM) and GLUT9 (inhibition of 60.25% at 50 μM). It exhibits analgesic and urate-lowering properties and is applicable for research in hyperuricemia and inflammatory pain.

Research Area

Metabolism Research, Pharmacology & Drug Discovery

Images & Validation

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Key Properties

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CAS Number	896584-55-7
MW	314.293
Formula	C₁₆H₁₄N₂O₅
SMILES	O=C(NC1=CC=C2OCOC2=C1)NC3=CC=C4OCCOC4=C3
Target	TRP/TRPV Channel,OAT,transporter,Cytochromes P450

Storage & Handling

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Storage	-20°C
Expiration Date	12 months from date of receipt.
Disclaimer	For research use only

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Gene Symbol

TRP/TRPV Channel,OAT,transporter,Cytochromes P450

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