Tianeptine Metabolite MC5 sodium

SKU: orb1980124

Description

MC5 is a bioactive β-oxidation metabolite of tianeptine that acts as a selective μ-opioid receptor (MOR) agonist, as demonstrated by BRET assays in HEK293T cells. Its MOR-dependent antidepressant-like efficacy is confirmed in vivo, reducing immobility in the mouse forced swim test at 30 mg/kg. This compound is a valuable research tool for studying MOR-mediated neuropharmacology and depression mechanisms.

Research Area

Metabolism Research, Pharmacology & Drug Discovery

Key Properties

• CAS Number: 115220-11-6
• MW: 430.88
• Formula: C₁₉H₂₀ClN₂O₄S.Na
• SMILES: O=C(CCCCNC1C2=C(N(S(=O)(C3=CC(Cl)=CC=C31)=O)C)C=CC=C2)[O-].[Na+]
• Target: Drug Metabolite

Storage & Handling

• Storage: -20°C
• Expiration Date: 12 months from date of receipt.
• Disclaimer: For research use only

Compound Identifiers

PubChem CID

46783084