Theliatinib tartrate

SKU: orb1744907

Description

Theliatinib tartrate is a potent, orally active, and highly selective ATP-competitive EGFR inhibitor, with a K_i of 0.05 nM. It shows strong activity against EGFR T790M/L858R mutants and >50-fold selectivity over other kinases, making it a valuable tool for in vitro and in vivo cancer research targeting EGFR-driven pathways.

Research Area

Cardiovascular Research, Signal Transduction

Key Properties

• CAS Number: 2413487-72-4
• MW: 592.6
• Formula: C₂₉H₃₂N₆O₈
• SMILES: [C@@H]([C@H](C(O)=O)O)(C(O)=O)O.N(C=1C2=C(C=C(OC)C(NC(=O)N3C[C@]4([C@@](C3)(CCN4C)[H])[H])=C2)N=CN1)C5=CC(C#C)=CC=C5
• Target: EGFR,Others

Storage & Handling

• Storage: -20°C
• Expiration Date: 12 months from date of receipt.
• Disclaimer: For research use only

Compound Identifiers

PubChem CID

168006833