TGR5 Receptor Agonist 3

• Catalog Number: orb1686487
• Category: Small Molecules
• Description: TGR5 Receptor Agonist 3
• CAS Number: 2643391-08-4
• Purity: 98%
• MW: 513.54
• SMILES: O=C(OCOCC)C1=COC=2C=CC(OC=3C=CN=CC3C(=O)N4C=5C=CC=CC5N(CC4)C6CC6)=CC21
• Formula: C₂₉H₂₇N₃O₆
• Biological Activity: TGR5 Receptor Agonist 3 is a G protein-coupled bile acid receptor 1 (GPBAR1, TGR5) agonist soft drug compound that decreases gallbladder filling, exhibits good gallbladder safety, and is able to act on hTGR5 (EC50: 16.4 nM) and mTGR5 (EC50: 209 nM).
• Note: For research use only
• Expiration Date: 12 months from date of receipt.