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TGR5 Receptor Agonist 3

TGR5 Receptor Agonist 3

Catalog Number: orb1686487

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Catalog Numberorb1686487
CategorySmall Molecules
DescriptionTGR5 Receptor Agonist 3
Purity98.00%
MW513.54
Biological ActivityTGR5 Receptor Agonist 3 is a G protein-coupled bile acid receptor 1 (GPBAR1, TGR5) agonist soft drug compound that decreases gallbladder filling, exhibits good gallbladder safety, and is able to act on hTGR5 (EC50: 16.4 nM) and mTGR5 (EC50: 209 nM).
CAS Number2643391-08-4
FormulaC29H27N3O6
SMILESC(=O)(N1C=2C(N(CC1)C3CC3)=CC=CC2)C=4C(OC=5C=C6C(=CC5)OC=C6C(OCOCC)=O)=CC=NC4
Storage-20°C
NoteFor research use only
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