Tazemetostat HCl

SKU: orb1738892

Description

Tazemetostat HCl (EPZ-6438) is a potent, selective, and orally available EZH2 inhibitor. It induces apoptosis and differentiation in SMARCB1-deleted malignant rhabdoid tumor (MRT) cells and causes tumor regression in mouse xenograft models, demonstrating therapeutic potential for EZH2-dependent cancers in preclinical research.

Research Area

Pharmacology & Drug Discovery

Key Properties

• CAS Number: 1467052-84-1
• MW: 609.21
• Formula: C₃₄H₄₅ClN₄O₄
• SMILES: Cl.CCN(C1CCOCC1)c1cc(cc(C(=O)NCc2c(C)cc(C)[nH]c2=O)c1C)-c1ccc(CN2CCOCC2)cc1
• Target: Others

Storage & Handling

• Storage: -20°C
• Expiration Date: 12 months from date of receipt.
• Disclaimer: For research use only

Compound Identifiers

PubChem CID

91617699