Queen's Award Received in 2021 ISO 9001 Certified Delivered over 1,000,000 bio-reagents to life science researchers Trusted by Life Science Communities
Cart summary

You have no items in your shopping cart.

Tariquidar

SKU: orb1225719

Description

A potent, specific P-gp inhibitor with Kd of 5.1 nM; potentiates the cytotoxicity of several drugs including doxorubicin, paclitaxel, etoposide, and vincristine in a panel of human MDR cell lines at 25-80 nM; exhibits potent i.v. and p.o. activity without apparently enhancing the plasma pharmacokinetics of paclitaxel or the toxicity of coadministered drugs.Breast Cancer Phase 2 Discontinued.

Images & Validation

Key Properties

CAS Number206873-63-4
MW646.7315
Purity>98% (HPLC)
FormulaC38H38N4O6
SMILESCOC1=CC2=C(CN(CCC3=CC=C(NC(=O)C4=C(NC(=O)C5=CC6=CC=CC=C6N=C5)C=C(OC)C(OC)=C4)C=C3)CC2)C=C1OC |c:17,26,28,31,40,43,49,t:2,4,10,12,22,24,34|
TargetP-glycoprotein
SolubilityDMSO: ≥ 100 mg/mL

Storage & Handling

StorageStorage temperature: -20°C. Stability: ≥ 2 years
Expiration Date12 months from date of receipt.
DisclaimerFor research use only

Alternative Names

XR 9576 | XR-9576 | XR9576

Similar Products

  • Tariquidar methanesulfonate hydrate [orb611537]

    >98%

    625375-83-9

    892.9887

    C40H52N4O15S2

    100 mg, 250 mg, 1 g
  • Tariquidar [orb1300901]

    >99.99% (May vary between batches)

    206873-63-4

    646.73

    C38H38N4O6

    100 mg, 5 mg, 10 mg, 25 mg, 50 mg
  • Tariquidar methanesulfonate hydrate [orb1708409]

    98.13% (May vary between batches)

    625375-83-9

    947.04

    C40H58N4O18S2

    2 mg
  • Tariquidar dimesylate [orb1687163]

    625375-84-0

    1695.9

    C80H94N8O25S4

    25 mg
  • Tariquidar dihydrochloride [orb1745075]

    1992047-62-7

    719.65

    C38H40Cl2N4O6

    100 mg, 250 mg, 1 g
Quality Guarantee

Quality Guarantee

Explore bioreagents carefree to elevate your research. All our products are rigorously tested for performance. If a product does not perform as described on its datasheet, our scientific support team will provide expert troubleshooting, a prompt replacement, or a refund. For full details, please see our Terms & Conditions and Buying Guide. Contact us at [email protected].

Protocol Information

Available Sizes

Select a size below

200 mg
500 mg
5 mg
$ 90.00
10 mg
$ 140.00
25 mg
$ 220.00
50 mg
$ 390.00
100 mg
$ 630.00