SSTR5 antagonist 4

SKU: orb3174920

Description

SSTR5 antagonist4 (compound 1) is a potent, highly selective, and orally bioavailable antagonist of somatostatin subtype 5 (SSTR5) with an hSSTR5 IC50 of 1.3 nM and an mSSTR5 IC50 of 1.0 nM. It has demonstrated effectiveness in oral glucose tolerance tests (OGTT) in high-fat diet (HFD) mice and is applicable in research related to type 2 diabetes.

Research Area

Pharmacology & Drug Discovery

Key Properties

• CAS Number: 916338-03-9
• MW: 491.61
• Formula: C₂₉H₃₄FN₃O₃
• SMILES: O=C(NC1CCN(CC2=CC(OCC)=C(C(OCC)=C2)C=3C=CC(F)=CC3)CC1)C4=CN=CC(=C4)C
• Target: Somatostatin

Storage & Handling

• Storage: -20°C
• Expiration Date: 12 months from date of receipt.
• Disclaimer: For research use only

Quick Database Links

Gene Symbol

Somatostatin