SRX3212

SKU: orb1739949

Description

SRX3212 is a potent dual BRD4/PI3Kα inhibitor, exhibiting IC50 values of 3.7 nM (BRD4 BD1) and 22 nM (PI3Kα). This novel small molecule is a significantly more potent BRD4 inhibitor than SF2523 and is a useful chemical probe for oncology research, particularly in studies of transcriptional regulation and PI3K signaling pathways in cancer models.

Key Properties

• CAS Number: 2735720-80-4
• MW: 505.54
• Formula: C₂₆H₂₃N₃O₆S
• SMILES: O=C1C2=C(C(=CS2)C3=CC(C(NCC=4C=CC=NC4)=O)=C5C(=C3)OCCO5)OC(=C1)N6CCOCC6
• Target: Others

Storage & Handling

• Storage: -20°C
• Expiration Date: 12 months from date of receipt.
• Disclaimer: For research use only

Compound Identifiers

PubChem CID

154571991