SR-12062

• Catalog Number: orb2814887
• Category: Small Molecules
• Description: SR-12062 functions as a full agonist at neurotensin receptor 1 (NTSR1), demonstrating notable efficacy and increased potency. Its EC50 value on NTSR1 is 2 μM, with complete receptor activation (Emax=100%). Compared to the parent compound 1 (EC50=178 μM; Emax=17%), SR-12062 shows approximately 90-fold greater potency.
• MW: 415.48
• CAS Number: 1623019-77-1
• Formula: C₂₅H₂₅N₃O₃
• SMILES: C(C(N[C@@H](CC(C)C)C(O)=O)=O)N1C=2C(=CC(=CC2)C3=CC4=C(N=C3)C=CC=C4)C=C1
• Storage: -20°C
• Note: For research use only