SB 271046 hydrochloride

SKU: orb1303142

Description

SB 271046 hydrochloride

Research Area

Neuroscience, Pharmacology & Drug Discovery

Key Properties

• CAS Number: 209481-24-3
• MW: 488.45
• Purity: 99.77%
• Formula: C₂₀H₂₂ClN₃O₃S₂·HCl
• SMILES: Cl.C[C@@H](CN1CC(=O)NC(=O)C1)N1CC(=O)NC(=O)C1
• Target: 5-HT Receptor
• Solubility: DMSO:45 mg/mL (92.13 mM);10% DMSO+40% PEG300+5% Tween 80+45% Saline:2 mg/mL (4.09 mM)

Bioactivity

• Target IC50:
  5-HT1D receptor:6.55 (pKi)|5-HT1A receptor:6.35 (pKi)|5-HT7 receptor:5.39 (pKi)|5-HT1B receptor:6.05 (pKi)|5-HT6:8.92(pKi)|5-HT2A receptor:5.62 (pKi)|5-HT2C receptor (human):5.73 (pKi)|5-HT1F receptor:5.95 (pKi)|5-HT4 receptor:5.27 (pKi)|5-HT2B receptor:5.41 (pKi)|5-HT1E:<4.99 (pKi)

Storage & Handling

• Storage: Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature.
• Expiration Date: 12 months from date of receipt.
• Disclaimer: For research use only

Alternative Names

channels, anticonvulsant, 5HT Receptor, 5-HT Receptor, 5-HT6, 5HTReceptor, 5-hydroxytryptamine Receptor, Inhibitor, inhibit, oral, MEST, selective, Serotonin Receptor, SB 271046, SB 271046 Hydrochloride, SB 271046 hydrochloride, SB 271046A, SB271046, SB-271046, SB271046 Hydrochloride, SB-271046 Hydrochloride, test

Compound Identifiers

PubChem CID

6918223