(S)-BI 2536

SKU: orb2564725

Description

(S)-BI 2536 is the less active enantiomer of the dual PLK1/BRD4 inhibitor BI 2536, exhibiting Ki values of 0.42 nM and 54 nM, respectively. This compound is a valuable chemical tool for probing kinase and bromodomain biology in cancer research, utilized in both in vitro biochemical assays and cellular studies.

Key Properties

• CAS Number: 1241725-90-5
• MW: 521.65
• Formula: C₂₈H₃₉N₇O₃
• SMILES: C(C)[C@@H]1N(C=2C(N(C)C1=O)=CN=C(NC3=C(OC)C=C(C(NC4CCN(C)CC4)=O)C=C3)N2)C5CCCC5

Storage & Handling

• Storage: -20°C
• Expiration Date: 12 months from date of receipt.
• Disclaimer: For research use only

Compound Identifiers

PubChem CID

86295201