RJG-2051

SKU: orb3028333

Description

RJG-2051 is a selective covalent inhibitor of aldo-keto reductase family 1 member C3 (AKR1C3), with an IC50 value of 13 nM. It interferes with the metabolism of substrates such as androgens, estrogens, and prostaglandins through AKR1C3. RJG-2051 holds potential for cancer research.

Research Area

Metabolism Research

Key Properties

• CAS Number: 2851993-77-4
• MW: 509.62
• Formula: C₂₆H₃₁N₅O₄S
• SMILES: O=C(C1=CC=C(C=C1)S(=O)(=O)N2N=C(N=C2)C3CCCCC3)N4CCN(C=5C=CC=CC5OC)CC4
• Target: Reductase

Storage & Handling

• Storage: -20°C
• Expiration Date: 12 months from date of receipt.
• Disclaimer: For research use only

Quick Database Links

Gene Symbol

Reductase